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Compound
PGDB_C029738
6 activity records1 related patents
2D structure
COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(CN6CCC7(CC6)Oc6ccc(C8CCC(=O)NC8=O)cc6O7)CC5)cc4)CC3)C[C@@H]2C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 4.98 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000741 | PGDB_C029738 | PGDB_AS000195 | View |
| IC50 | - | = | 0.00011 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A004860 | PGDB_C029738 | PGDB_AS000481 | View |
| % Degradation | - | = | 93 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A005874 | PGDB_C029738 | PGDB_AS001838 | View |
| % Degradation | - | = | 44 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079866 | PGDB_C029738 | PGDB_AS002463 | View |
| % Degradation | - | = | 79 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080228 | PGDB_C029738 | PGDB_AS002389 | View |
| % Degradation | - | = | 80 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A081051 | PGDB_C029738 | PGDB_AS001354 | View |