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Compound
PGDB_C029743
6 activity records1 related patents
2D structure
COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(C)(CN6CCC7(CC6)COc6cc(N8CCC(=O)NC8=O)ccc67)CC5)cc4)CC3)C[C@@H]2C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 48 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000040 | PGDB_C029743 | PGDB_AS002463 | View |
| % Degradation | - | = | 82 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A001389 | PGDB_C029743 | PGDB_AS002389 | View |
| % Degradation | - | = | 48 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A001787 | PGDB_C029743 | PGDB_AS001354 | View |
| % Degradation | - | = | 66 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A003143 | PGDB_C029743 | PGDB_AS001838 | View |
| IC50 | - | = | 0.051 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081144 | PGDB_C029743 | PGDB_AS000195 | View |
| IC50 | - | = | 0.012 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A081539 | PGDB_C029743 | PGDB_AS000481 | View |