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Compound
PGDB_C029745
6 activity records1 related patents
2D structure
COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(C(=O)N4CCC(CN5CCC6(CCc7ccc(N8CCC(=O)NC8=O)cc7O6)CC5)CC4)cc3)C2(C)C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 29 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000769 | PGDB_C029745 | PGDB_AS002389 | View |
| IC50 | - | < | 0.000026 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A001449 | PGDB_C029745 | PGDB_AS000481 | View |
| % Degradation | - | = | 20 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A003183 | PGDB_C029745 | PGDB_AS001838 | View |
| % Degradation | - | = | 17 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A003925 | PGDB_C029745 | PGDB_AS002463 | View |
| % Degradation | - | = | 17 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A004394 | PGDB_C029745 | PGDB_AS001354 | View |
| IC50 | - | = | 8.89 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079920 | PGDB_C029745 | PGDB_AS000195 | View |