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Compound
PGDB_C029773
5 activity records1 related patents
2D structure
C[C@@H]1N(c2ccc(C#N)c(Cl)c2)CCC12CCN(c1ccc(C(=O)N3CCC(O[C@H]4C[C@H](CN5CCN6c7ccc(N8CCC(=O)NC8=O)cc7OCC[C@H]6C5)C4)CC3)cc1)CC2Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 67 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000612 | PGDB_C029773 | PGDB_AS001354 | View |
| % Degradation | - | = | 93 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A002899 | PGDB_C029773 | PGDB_AS002389 | View |
| IC50 | - | = | 0.009 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A003917 | PGDB_C029773 | PGDB_AS000271 | View |
| % Degradation | - | = | 74 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A003987 | PGDB_C029773 | PGDB_AS002463 | View |
| % Degradation | - | = | 80 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A004861 | PGDB_C029773 | PGDB_AS001838 | View |