Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C029779
5 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(O[C@H]5CC[C@@H](CN6CCC7(CCc8ccc(N9CCC(=O)NC9=O)cc8O7)CC6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(C(F)(F)F)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.093 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A000376 | PGDB_C029779 | PGDB_AS000271 | View |
| % Degradation | - | = | 14 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A005218 | PGDB_C029779 | PGDB_AS001354 | View |
| % Degradation | - | = | 3 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078824 | PGDB_C029779 | PGDB_AS002463 | View |
| % Degradation | - | = | 54 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079168 | PGDB_C029779 | PGDB_AS002389 | View |
| % Degradation | - | = | 64 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A080670 | PGDB_C029779 | PGDB_AS001838 | View |