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Compound
PGDB_C029792
6 activity records1 related patents
2D structure
COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(C)(CN6CCC7(CC6)Cc6ccc(N8CCC(=O)NC8=O)cc6O7)CC5)cc4)CC3)C[C@@H]2C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.014 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A000928 | PGDB_C029792 | PGDB_AS000481 | View |
| % Degradation | - | = | 85 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A001668 | PGDB_C029792 | PGDB_AS001838 | View |
| % Degradation | - | = | 44 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A004672 | PGDB_C029792 | PGDB_AS002463 | View |
| % Degradation | - | = | 81 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A005022 | PGDB_C029792 | PGDB_AS002389 | View |
| % Degradation | - | = | 56 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A079297 | PGDB_C029792 | PGDB_AS001354 | View |
| IC50 | - | = | 0.38 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080477 | PGDB_C029792 | PGDB_AS000195 | View |