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Compound
PGDB_C029802
6 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CC5)COc5cc(N7CCC(=O)NC7=O)ccc56)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 86 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000295 | PGDB_C029802 | PGDB_AS002463 | View |
| % Degradation | - | = | 75 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A002286 | PGDB_C029802 | PGDB_AS001354 | View |
| IC50 | - | = | 0.006 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A078139 | PGDB_C029802 | PGDB_AS000481 | View |
| % Degradation | - | = | 93 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079946 | PGDB_C029802 | PGDB_AS002389 | View |
| % Degradation | - | = | 87 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A080128 | PGDB_C029802 | PGDB_AS001838 | View |
| IC50 | - | = | 0.082 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080202 | PGDB_C029802 | PGDB_AS000195 | View |