Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C029811
6 activity records1 related patents
2D structure
N#Cc1ccc(N[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7ccc(N8CCC(=O)NC8=O)cc7OCC[C@H]6C5)CC4)cc3)CC2)cc1ClCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 87 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000275 | PGDB_C029811 | PGDB_AS001838 | View |
| % Degradation | - | = | 50 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A001508 | PGDB_C029811 | PGDB_AS002463 | View |
| % Degradation | - | = | 84 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A001993 | PGDB_C029811 | PGDB_AS001354 | View |
| % Degradation | - | = | 54 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078028 | PGDB_C029811 | PGDB_AS002389 | View |
| IC50 | - | = | 0.003 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A079053 | PGDB_C029811 | PGDB_AS000271 | View |
| IC50 | - | = | 0.098 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080535 | PGDB_C029811 | PGDB_AS000195 | View |