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Compound
PGDB_C029831
6 activity records1 related patents
2D structure
CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN5c6ccc(N7CCC(=O)NC7=O)cc6OCC[C@H]5C4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 80 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000406 | PGDB_C029831 | PGDB_AS001354 | View |
| % Degradation | - | = | 90 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000621 | PGDB_C029831 | PGDB_AS001838 | View |
| % Degradation | - | = | 71 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A003520 | PGDB_C029831 | PGDB_AS002389 | View |
| % Degradation | - | = | 32 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A005446 | PGDB_C029831 | PGDB_AS002463 | View |
| IC50 | - | = | 0.0015 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A005645 | PGDB_C029831 | PGDB_AS000481 | View |
| IC50 | - | = | 0.11 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079503 | PGDB_C029831 | PGDB_AS000195 | View |