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Compound
PGDB_C029840
5 activity records1 related patents
2D structure
COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(O[C@H]6CC[C@@H](CN7CCN8c9ccc(N%10CCC(=O)NC%10=O)cc9OCC[C@H]8C7)CC6)CC5)c(F)c4)CC3)C[C@@H]2C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 51 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000086 | PGDB_C029840 | PGDB_AS001838 | View |
| % Degradation | - | = | 30 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A001953 | PGDB_C029840 | PGDB_AS002463 | View |
| % Degradation | - | = | 5 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A005235 | PGDB_C029840 | PGDB_AS001354 | View |
| IC50 | - | = | 0.14 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A080540 | PGDB_C029840 | PGDB_AS000271 | View |
| % Degradation | - | = | 68 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081044 | PGDB_C029840 | PGDB_AS002389 | View |