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Compound
PGDB_C029887
6 activity records1 related patents
2D structure
O=C1CCN(c2ccc3c(c2)OC2(CCN(CC4CCNCC4)CC2)C3)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.043 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000141 | PGDB_C029887 | PGDB_AS000195 | View |
| % Degradation | - | = | 48 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A003085 | PGDB_C029887 | PGDB_AS001838 | View |
| % Degradation | - | = | 48 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078010 | PGDB_C029887 | PGDB_AS002463 | View |
| IC50 | - | = | 0.12 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A078157 | PGDB_C029887 | PGDB_AS000481 | View |
| % Degradation | - | = | 56 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078338 | PGDB_C029887 | PGDB_AS001354 | View |
| % Degradation | - | = | 52 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081463 | PGDB_C029887 | PGDB_AS002389 | View |