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Compound
PGDB_C029897
6 activity records1 related patents
2D structure
CN(c1ccc2c(c1)OCC21CCN(CC2CCN(c3ccc(C(=O)N[C@H]4CC[C@H](Oc5ccc(C#N)c(Cl)c5)CC4)nn3)CC2)CC1)C1CCC(=O)NC1=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 33 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000087 | PGDB_C029897 | PGDB_AS002463 | View |
| % Degradation | - | = | 77 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000438 | PGDB_C029897 | PGDB_AS001838 | View |
| IC50 | - | = | 1.41 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A002838 | PGDB_C029897 | PGDB_AS000481 | View |
| IC50 | - | = | 0.94 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A005480 | PGDB_C029897 | PGDB_AS000195 | View |
| % Degradation | - | = | 56 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078889 | PGDB_C029897 | PGDB_AS002389 | View |
| % Degradation | - | = | 61 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078966 | PGDB_C029897 | PGDB_AS001354 | View |