Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C029903
5 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC5(CC(N6CCN7c8ccc(N9CCC(=O)NC9=O)cc8OCC[C@H]7C6)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.008 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A000253 | PGDB_C029903 | PGDB_AS000271 | View |
| % Degradation | - | = | 81 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000829 | PGDB_C029903 | PGDB_AS001354 | View |
| % Degradation | - | = | 92 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A004144 | PGDB_C029903 | PGDB_AS001838 | View |
| % Degradation | - | = | 89 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078715 | PGDB_C029903 | PGDB_AS002389 | View |
| % Degradation | - | = | 70 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081036 | PGDB_C029903 | PGDB_AS002463 | View |