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Compound
PGDB_C029918
5 activity records1 related patents
2D structure
COc1cc2c(c3c1C1(CCN(CC4CCN(c5ccc(N6CCC7(CC6)C[C@H](C)N(c6ccc(C#N)c(Cl)c6)C7)cc5)CC4)CC1)CO3)CN([C@H]1CCC(=O)NC1=O)C2=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 90 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000058 | PGDB_C029918 | PGDB_AS001838 | View |
| IC50 | - | = | 0.008 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A002107 | PGDB_C029918 | PGDB_AS000271 | View |
| % Degradation | - | = | 45 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A005367 | PGDB_C029918 | PGDB_AS002463 | View |
| % Degradation | - | = | 65 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080008 | PGDB_C029918 | PGDB_AS002389 | View |
| % Degradation | - | = | 91 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A081440 | PGDB_C029918 | PGDB_AS001354 | View |