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Compound
PGDB_C029959
6 activity records1 related patents
2D structure
Cc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(OC6CCC(CN7CCN8c9cc(N[C@H]%10CCC(=O)NC%10=O)ccc9OCC[C@H]8C7)CC6)CC5)cc4F)CC3)C[C@@H]2C)cc(C)c1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 40 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000049 | PGDB_C029959 | PGDB_AS002389 | View |
| IC50 | - | = | 0.83 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A000448 | PGDB_C029959 | PGDB_AS000271 | View |
| % Degradation | - | = | 7 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A004196 | PGDB_C029959 | PGDB_AS002463 | View |
| % Degradation | - | = | 20 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A006482 | PGDB_C029959 | PGDB_AS001838 | View |
| % Degradation | - | = | 13 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078962 | PGDB_C029959 | PGDB_AS001354 | View |
| IC50 | - | = | 7.2 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080902 | PGDB_C029959 | PGDB_AS000195 | View |