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Compound
PGDB_C029961
6 activity records1 related patents
2D structure
C[C@H]1CN(c2ccc(C#N)c(Cl)c2)CC12CCN(c1ccc(C(=O)N3CCC(CN4CCN5c6ccc(C7CCC(=O)NC7=O)cc6OCC[C@H]5C4)CC3)nn1)CC2Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 93 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000423 | PGDB_C029961 | PGDB_AS001354 | View |
| % Degradation | - | = | 85 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A002679 | PGDB_C029961 | PGDB_AS002463 | View |
| % Degradation | - | = | 87 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A003004 | PGDB_C029961 | PGDB_AS002389 | View |
| IC50 | - | < | 0.014 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A005650 | PGDB_C029961 | PGDB_AS000195 | View |
| IC50 | - | = | 0.008 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A006219 | PGDB_C029961 | PGDB_AS000271 | View |
| % Degradation | - | = | 92 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078051 | PGDB_C029961 | PGDB_AS001838 | View |