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Compound
PGDB_C029969
5 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCC6(CC5)COc5c6cc(Cl)c6c5CN([C@H]5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 94 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000117 | PGDB_C029969 | PGDB_AS001838 | View |
| IC50 | - | = | 0.027 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A002635 | PGDB_C029969 | PGDB_AS000271 | View |
| % Degradation | - | = | 90 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A004636 | PGDB_C029969 | PGDB_AS001354 | View |
| % Degradation | - | = | 40 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080177 | PGDB_C029969 | PGDB_AS002463 | View |
| % Degradation | - | = | 72 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081570 | PGDB_C029969 | PGDB_AS002389 | View |