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Compound
PGDB_C029979
10 activity records1 related patents
2D structure
COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCN6c7ccc(N8CCC(=O)NC8=O)cc7OCC[C@H]6C4)C5)cc3)C2(C)C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 90 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000068 | PGDB_C029979 | PGDB_AS001838 | View |
| % Degradation | - | = | 81 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000070 | PGDB_C029979 | PGDB_AS002463 | View |
| % Degradation | - | = | 81 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A001985 | PGDB_C029979 | PGDB_AS002463 | View |
| % Degradation | - | = | 90 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A002211 | PGDB_C029979 | PGDB_AS001838 | View |
| % Degradation | - | = | 86 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A002832 | PGDB_C029979 | PGDB_AS002389 | View |
| % Degradation | - | = | 84 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A005387 | PGDB_C029979 | PGDB_AS001354 | View |
| % Degradation | - | = | 84 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078666 | PGDB_C029979 | PGDB_AS001354 | View |
| IC50 | - | = | 0.004 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A079224 | PGDB_C029979 | PGDB_AS000271 | View |
| IC50 | - | = | 0.004 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A080814 | PGDB_C029979 | PGDB_AS000271 | View |
| % Degradation | - | = | 86 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081875 | PGDB_C029979 | PGDB_AS002389 | View |