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Compound
PGDB_C030016
6 activity records1 related patents
2D structure
Cc1cc(C(=O)N2CCC(CN3CCN4c5cc(N[C@H]6CCC(=O)NC6=O)ccc5OCC[C@H]4C3)CC2)ccc1N1CCC2(CC1)C[C@H](C)N(c1ccc(C#N)c(Cl)c1)C2Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 79 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000369 | PGDB_C030016 | PGDB_AS002389 | View |
| IC50 | - | = | 0.33 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A001761 | PGDB_C030016 | PGDB_AS000195 | View |
| % Degradation | - | = | 53 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A004020 | PGDB_C030016 | PGDB_AS002463 | View |
| IC50 | - | = | 0.033 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A004533 | PGDB_C030016 | PGDB_AS000271 | View |
| % Degradation | - | = | 85 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A080598 | PGDB_C030016 | PGDB_AS001838 | View |
| % Degradation | - | = | 18 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A081526 | PGDB_C030016 | PGDB_AS001354 | View |