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Compound
PGDB_C030021
6 activity records1 related patents
2D structure
COc1cc(N2CC3(CCN(c4ncc(C(=O)N5CCC6(CCC(N7CCN8c9cc(N[C@H]%10CCC(=O)NC%10=O)ccc9OCC[C@H]8C7)C6)CC5)cn4)CC3)C[C@@H]2C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 55 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000089 | PGDB_C030021 | PGDB_AS002463 | View |
| % Degradation | - | = | 58 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000783 | PGDB_C030021 | PGDB_AS001354 | View |
| IC50 | - | = | 0.061 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A002796 | PGDB_C030021 | PGDB_AS000271 | View |
| % Degradation | - | = | 83 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A005911 | PGDB_C030021 | PGDB_AS002389 | View |
| % Degradation | - | = | 75 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A006859 | PGDB_C030021 | PGDB_AS001838 | View |
| IC50 | - | = | 0.83 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078592 | PGDB_C030021 | PGDB_AS000195 | View |