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Compound
PGDB_C030026
6 activity records1 related patents
2D structure
COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC6(CC5)CC(N5CCN7c8ccc(N9CCC(=O)NC9=O)cc8OCC[C@H]7C5)C6)c(F)c4)CC3)C[C@@H]2C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 48 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000173 | PGDB_C030026 | PGDB_AS001354 | View |
| IC50 | - | = | 0.17 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000541 | PGDB_C030026 | PGDB_AS000195 | View |
| % Degradation | - | = | 77 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A001172 | PGDB_C030026 | PGDB_AS001838 | View |
| % Degradation | - | = | 81 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A005607 | PGDB_C030026 | PGDB_AS002389 | View |
| % Degradation | - | = | 54 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079422 | PGDB_C030026 | PGDB_AS002463 | View |
| IC50 | - | = | 0.008 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A080881 | PGDB_C030026 | PGDB_AS000271 | View |