Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C030029
6 activity records1 related patents
2D structure
COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(CN6CCN7c8cc(N[C@H]9CCC(=O)NC9=O)ccc8OCC[C@H]7C6)CC5)c(Cl)c4)CC3)C[C@@H]2C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 5.11 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000260 | PGDB_C030029 | PGDB_AS000195 | View |
| % Degradation | - | = | 83 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A001863 | PGDB_C030029 | PGDB_AS001838 | View |
| % Degradation | - | = | 77 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A002935 | PGDB_C030029 | PGDB_AS002389 | View |
| IC50 | - | = | 0.018 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A004895 | PGDB_C030029 | PGDB_AS000271 | View |
| % Degradation | - | = | 54 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078786 | PGDB_C030029 | PGDB_AS001354 | View |
| % Degradation | - | = | 48 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080488 | PGDB_C030029 | PGDB_AS002463 | View |