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Compound
PGDB_C030075
5 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(O[C@H]5CC[C@@H](CN6CCN7c8cc(N[C@H]9CCC(=O)NC9=O)ccc8OCC[C@H]7C6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(C(F)(F)F)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.4 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A000186 | PGDB_C030075 | PGDB_AS000271 | View |
| % Degradation | - | = | 14 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A001874 | PGDB_C030075 | PGDB_AS002463 | View |
| % Degradation | - | = | 25 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A004851 | PGDB_C030075 | PGDB_AS001838 | View |
| % Degradation | - | = | 40 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078654 | PGDB_C030075 | PGDB_AS002389 | View |