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Compound
PGDB_C030077
5 activity records1 related patents
2D structure
Cc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(CN6CCN7c8ccc(N9CCC(=O)NC9=O)cc8OCC[C@H]7C6)CC5)cc4F)CC3)C[C@@H]2C)cc(C)c1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 63 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A000578 | PGDB_C030077 | PGDB_AS001354 | View |
| % Degradation | - | = | 88 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A004911 | PGDB_C030077 | PGDB_AS002389 | View |
| % Degradation | - | = | 85 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A006070 | PGDB_C030077 | PGDB_AS001838 | View |
| % Degradation | - | = | 63 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078397 | PGDB_C030077 | PGDB_AS002463 | View |
| IC50 | - | = | 0.017 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A079816 | PGDB_C030077 | PGDB_AS000271 | View |