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Compound
PGDB_C030080
5 activity records1 related patents
2D structure
CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN5c6ccc(N7CCC(=O)NC7=O)cc6OCC[C@H]5C4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(C(F)(F)F)c1FCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 18 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000042 | PGDB_C030080 | PGDB_AS002463 | View |
| IC50 | - | = | 0.02 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A004403 | PGDB_C030080 | PGDB_AS000271 | View |
| % Degradation | - | = | 48 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A005830 | PGDB_C030080 | PGDB_AS001354 | View |
| % Degradation | - | = | 24 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A006648 | PGDB_C030080 | PGDB_AS002389 | View |
| % Degradation | - | = | 61 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A079901 | PGDB_C030080 | PGDB_AS001838 | View |