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Compound
PGDB_C030081
6 activity records1 related patents
2D structure
N#Cc1ccc(N2CC3(CCN(c4ccc(C(=O)N5CCC(CN6CCN7c8ccc(N9CCC(=O)NC9=O)cc8OCC[C@H]7C6)CC5)cc4)CC3)C[C@@H]2C(F)(F)F)cc1ClCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 79 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000565 | PGDB_C030081 | PGDB_AS002463 | View |
| % Degradation | - | = | 74 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A004362 | PGDB_C030081 | PGDB_AS001354 | View |
| IC50 | - | = | 0.004 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A079181 | PGDB_C030081 | PGDB_AS000271 | View |
| IC50 | - | = | 0.76 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080338 | PGDB_C030081 | PGDB_AS000195 | View |
| % Degradation | - | = | 91 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A081654 | PGDB_C030081 | PGDB_AS001838 | View |
| % Degradation | - | = | 94 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081740 | PGDB_C030081 | PGDB_AS002389 | View |