Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C030095
6 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(F)(CN5CCN6c7ccc(N8CCC(=O)NC8=O)cc7OCC[C@H]6C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1FCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 92 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000348 | PGDB_C030095 | PGDB_AS002389 | View |
| % Degradation | - | = | 91 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A006102 | PGDB_C030095 | PGDB_AS001838 | View |
| % Degradation | - | = | 88 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078111 | PGDB_C030095 | PGDB_AS001354 | View |
| IC50 | - | = | 0.001 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A078557 | PGDB_C030095 | PGDB_AS000271 | View |
| % Degradation | - | = | 81 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080952 | PGDB_C030095 | PGDB_AS002463 | View |
| IC50 | - | = | 0.087 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081574 | PGDB_C030095 | PGDB_AS000195 | View |