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Compound
PGDB_C030100
6 activity records1 related patents
2D structure
COC1(CN2CCN3c4ccc(N5CCC(=O)NC5=O)cc4OCC[C@H]3C2)CCN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3F)C4)nn2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.42 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000691 | PGDB_C030100 | PGDB_AS000195 | View |
| % Degradation | - | = | 94 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A003289 | PGDB_C030100 | PGDB_AS001838 | View |
| IC50 | - | = | 0.002 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A004517 | PGDB_C030100 | PGDB_AS000271 | View |
| % Degradation | - | = | 83 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079197 | PGDB_C030100 | PGDB_AS002463 | View |
| % Degradation | - | = | 91 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A079376 | PGDB_C030100 | PGDB_AS001354 | View |
| % Degradation | - | = | 86 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079988 | PGDB_C030100 | PGDB_AS002389 | View |