Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C030116
3 activity records1 related patents
2D structure
COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(C5CCC(=O)NC5=O)c5ccccc56)CC4)c(Cl)c3)C2(C)C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 21 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000073 | PGDB_C030116 | PGDB_AS002389 | View |
| % Degradation | - | = | 9 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A002476 | PGDB_C030116 | PGDB_AS002463 | View |
| IC50 | - | = | 28.86 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078923 | PGDB_C030116 | PGDB_AS000195 | View |