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Compound
PGDB_C030119
6 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(O[C@H]5CC[C@H](CN6CCN7c8ccc(N9CCC(=O)NC9=O)cc8OCC[C@H]7C6)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1FCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.19 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000081 | PGDB_C030119 | PGDB_AS000195 | View |
| % Degradation | - | = | 87 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A004463 | PGDB_C030119 | PGDB_AS002389 | View |
| IC50 | - | = | 0.001 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A006038 | PGDB_C030119 | PGDB_AS000271 | View |
| % Degradation | - | = | 84 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A006972 | PGDB_C030119 | PGDB_AS001838 | View |
| % Degradation | - | = | 85 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A080299 | PGDB_C030119 | PGDB_AS001354 | View |
| % Degradation | - | = | 80 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A081394 | PGDB_C030119 | PGDB_AS002463 | View |