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Compound
PGDB_C030124
6 activity records1 related patents
2D structure
N#Cc1ccc(N2CC3(CCN(c4ccc(C(=O)N5CCC(Cl)(CN6CCN7c8ccc(N9CCC(=O)NC9=O)cc8OCC[C@H]7C6)CC5)cc4)CC3)CC2C(F)(F)F)cc1ClCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 84 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000207 | PGDB_C030124 | PGDB_AS002389 | View |
| % Degradation | - | = | 65 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A006474 | PGDB_C030124 | PGDB_AS002463 | View |
| % Degradation | - | = | 87 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A006763 | PGDB_C030124 | PGDB_AS001838 | View |
| IC50 | - | = | 0.005 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A078391 | PGDB_C030124 | PGDB_AS000271 | View |
| IC50 | - | = | 1.33 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A080438 | PGDB_C030124 | PGDB_AS000195 | View |
| % Degradation | - | = | 84 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A081761 | PGDB_C030124 | PGDB_AS001354 | View |