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Compound
PGDB_C030130
6 activity records1 related patents
2D structure
COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7ccc(N8CCC(=O)NC8=O)cc7OCC[C@H]6C5)CC4)c(S(C)(=O)=O)c3)C2(C)C)ccc1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 91 | % | 100 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A000060 | PGDB_C030130 | PGDB_AS002389 | View |
| % Degradation | - | = | 86 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A002544 | PGDB_C030130 | PGDB_AS001354 | View |
| IC50 | - | = | 0.00047 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A005839 | PGDB_C030130 | PGDB_AS000271 | View |
| % Degradation | - | = | 85 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A005843 | PGDB_C030130 | PGDB_AS001838 | View |
| IC50 | - | = | 0.051 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079569 | PGDB_C030130 | PGDB_AS000195 | View |
| % Degradation | - | = | 73 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A079912 | PGDB_C030130 | PGDB_AS002463 | View |