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Nc1nnc(-c2ccccc2O)cc1N1CC2CCC(C1)N2c1ncc(C2CCN(Cc3cccc(N4CCC(=O)NC4=O)c3)CC2)cn1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | - | - | H2126 | WO2026061475A1 | PGDB_A000910 | PGDB_C030297 | PGDB_AS001417 | View | |
| IC50 | - | = | 700-900 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A001248 | PGDB_C030297 | PGDB_AS000282 | View | |
| % Inhibition | - | = | 70-80 | % | 2 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A003852 | PGDB_C030297 | PGDB_AS001031 | View | |
| % Inhibition | - | = | 30-40 | % | 0.5 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A004695 | PGDB_C030297 | PGDB_AS000662 | View | |
| IC50 | - | = | 30-50 | nM | - | — | - | - | H1944 | WO2026061475A1 | PGDB_A006534 | PGDB_C030297 | PGDB_AS001924 | View |