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O=C1CCN(c2ccc(CN3CCC(c4c[nH]c5nnc(-c6ccccc6O)cc45)CC3)c(F)c2)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 60-70 | % | 2 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A001826 | PGDB_C030429 | PGDB_AS001031 | View | |
| IC50 | - | = | 200-500 | nM | - | — | - | - | H2126 | WO2026061475A1 | PGDB_A004261 | PGDB_C030429 | PGDB_AS001417 | View | |
| IC50 | - | = | 1-5 | nM | - | — | - | - | BT549 | WO2026061475A1 | PGDB_A004688 | PGDB_C030429 | PGDB_AS002259 | View | |
| % Inhibition | - | = | 20-30 | % | 0.5 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A078072 | PGDB_C030429 | PGDB_AS000662 | View | |
| IC50 | - | = | 20-30 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A081742 | PGDB_C030429 | PGDB_AS000282 | View |