Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C030460
4 activity records1 related patents
2D structure
Nc1nnc(-c2cc(F)ccc2O)cc1N1CC2CCC(C1)N2CCc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | <= | 50 | % | Concentration series: 500 nM, 50 nM | - | SMARCA2 | - | MV-4-11 | WO2026061475A1 | PGDB_A000287 | PGDB_C030460 | PGDB_AS002335 | View |
| % Degradation | - | <= | 50 | % | Concentration series: 500 nM, 50 nM | - | SMARCA4 | - | MV-4-11 | WO2026061475A1 | PGDB_A004659 | PGDB_C030460 | PGDB_AS002340 | View |
| % Inhibition | - | = | 60-70 | % | 2 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A004758 | PGDB_C030460 | PGDB_AS001031 | View |
| % Inhibition | - | = | 30-40 | % | 0.5 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A081178 | PGDB_C030460 | PGDB_AS000662 | View |