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CC1(NS(=O)(=O)c2cc(N3CCN(c4ccc(C5CCC(=O)NC5=O)c(F)c4)CC3)c3cnc(-c4nnc(C(F)F)s4)n3c2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 1.25 | uM | - | — | PARG | - | NCIH-460 | WO2026062066A1 | PGDB_A005288 | PGDB_C030608 | PGDB_AS002426 | View | |
| IC50 | - | = | 0.053 | uM | - | — | PARG | - | - | WO2026062066A1 | PGDB_A006645 | PGDB_C030608 | PGDB_AS002282 | View | |
| EC50 | - | > | 20 | uM | - | — | PARG | - | U2OS | WO2026062066A1 | PGDB_A079874 | PGDB_C030608 | PGDB_AS002468 | View |