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SIMM · NJU
Assay
PGDB_AS002426
System: cell_based
Cell line: NCIH-460
Assay context summary
Assay context
19 activity records
Assay family
viability
System
cell_based
Readout
EC50
E3
Not specified
Cell line
NCIH-460
Organism
Homo sapiens
Activity compounds and values
Activity records
19 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.633
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A000600
PGDB_C030613
PGDB_AS002426
View
EC50
-
=
1.25
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A001019
PGDB_C030622
PGDB_AS002426
View
EC50
-
=
0.07
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A002392
PGDB_C030612
PGDB_AS002426
View
EC50
-
>
20
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A002572
PGDB_C030606
PGDB_AS002426
View
EC50
-
>
12.46
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A003474
PGDB_C030621
PGDB_AS002426
View
EC50
-
>
20
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A004033
PGDB_C030605
PGDB_AS002426
View
EC50
-
=
1.33
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A004520
PGDB_C030610
PGDB_AS002426
View
EC50
-
>
20
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A004835
PGDB_C025567
PGDB_AS002426
View
EC50
-
=
1.25
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A005288
PGDB_C030608
PGDB_AS002426
View
EC50
-
=
4.169
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A005378
PGDB_C030617
PGDB_AS002426
View
EC50
-
>
20
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A005677
PGDB_C030618
PGDB_AS002426
View
EC50
-
=
0.596
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A078081
PGDB_C030611
PGDB_AS002426
View
EC50
-
>
12.57
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A078355
PGDB_C030616
PGDB_AS002426
View
EC50
-
=
14.96
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A078356
PGDB_C030615
PGDB_AS002426
View
EC50
-
=
0.643
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A078498
PGDB_C030624
PGDB_AS002426
View
EC50
-
=
1.023
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A078524
PGDB_C030609
PGDB_AS002426
View
EC50
-
=
1.16
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A078968
PGDB_C030625
PGDB_AS002426
View
EC50
-
>
7.22
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A079173
PGDB_C030620
PGDB_AS002426
View
EC50
-
>
18.3
uM
-
—
PARG
-
NCIH-460
WO2026062066A1
PGDB_A080856
PGDB_C030607
PGDB_AS002426
View