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SIMM · NJU
Assay
PGDB_AS002282
System: biochemical
Assay context summary
Assay context
43 activity records
Assay family
biochemical
System
biochemical
Readout
IC50
E3
Not specified
Activity compounds and values
Activity records
43 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
0.114
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A000487
PGDB_C025567
PGDB_AS002282
View
IC50
-
=
0.079
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A000839
PGDB_C030642
PGDB_AS002282
View
IC50
-
=
0.148
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A000848
PGDB_C030643
PGDB_AS002282
View
IC50
-
=
0.144
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A000894
PGDB_C030646
PGDB_AS002282
View
IC50
-
=
5.5
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A001164
PGDB_C030630
PGDB_AS002282
View
IC50
-
=
0.716
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A001205
PGDB_C030648
PGDB_AS002282
View
IC50
-
=
16
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A002057
PGDB_C030633
PGDB_AS002282
View
IC50
-
=
1
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A002096
PGDB_C030621
PGDB_AS002282
View
IC50
-
=
0.1
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A002239
PGDB_C030635
PGDB_AS002282
View
IC50
-
=
0.146
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A002347
PGDB_C030607
PGDB_AS002282
View
IC50
-
=
0.207
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A002859
PGDB_C030637
PGDB_AS002282
View
IC50
-
=
0.17
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A003037
PGDB_C030622
PGDB_AS002282
View
IC50
-
=
0.347
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A003349
PGDB_C030641
PGDB_AS002282
View
IC50
-
=
0.074
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A003377
PGDB_C030645
PGDB_AS002282
View
IC50
-
=
0.167
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A003496
PGDB_C030613
PGDB_AS002282
View
IC50
-
=
0.25
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A003498
PGDB_C030639
PGDB_AS002282
View
IC50
-
=
0.093
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A003707
PGDB_C030612
PGDB_AS002282
View
IC50
-
=
0.394
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A004807
PGDB_C030617
PGDB_AS002282
View
IC50
-
>
20
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A004870
PGDB_C030634
PGDB_AS002282
View
IC50
-
=
0.697
uM
-
—
PARG
-
-
WO2026062066A1
PGDB_A004898
PGDB_C030619
PGDB_AS002282
View