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C[C@H]1CN(c2cc(S(=O)(=O)NC3(C)CC3)cn3c(-c4nnc(C(F)F)s4)ncc23)C[C@H](O)N1C(=O)NCCCCCCCOc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.633 | uM | - | — | PARG | - | NCIH-460 | WO2026062066A1 | PGDB_A000600 | PGDB_C030613 | PGDB_AS002426 | View | |
| EC50 | - | > | 20 | uM | - | — | PARG | - | U2OS | WO2026062066A1 | PGDB_A000965 | PGDB_C030613 | PGDB_AS002468 | View | |
| IC50 | - | = | 0.167 | uM | - | — | PARG | - | - | WO2026062066A1 | PGDB_A003496 | PGDB_C030613 | PGDB_AS002282 | View |