Assay

PGDB_AS000831

System: cell_basedTarget: VAV1Cell line: 293T-VAV1-FLAG
Assay context summary

Assay context

55 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetVAV1
E3Not specified
Cell line293T-VAV1-FLAG
OrganismHomo sapiens
Detection targetprotein_degradation
Activity compounds and values

Activity records

55 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031440
DC50-=45.09nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A000063PGDB_C031440PGDB_AS000831View
2D structure for PGDB_C031456
DC50-=13.11nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A000064PGDB_C031456PGDB_AS000831View
2D structure for PGDB_C031416
DC50-=9.04nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A000510PGDB_C031416PGDB_AS000831View
2D structure for PGDB_C029470
DC50-=31.86nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A000709PGDB_C029470PGDB_AS000831View
2D structure for PGDB_C031427
DC50-=3.8nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A000756PGDB_C031427PGDB_AS000831View
2D structure for PGDB_C031451
DC50-=15.61nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A000933PGDB_C031451PGDB_AS000831View
2D structure for PGDB_C031415
DC50-=1.69nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A001222PGDB_C031415PGDB_AS000831View
2D structure for PGDB_C031413
DC50-=11.57nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A001920PGDB_C031413PGDB_AS000831View
2D structure for PGDB_C031417
DC50-=15.82nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A001996PGDB_C031417PGDB_AS000831View
2D structure for PGDB_C031445
DC50-=26.47nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A002046PGDB_C031445PGDB_AS000831View
2D structure for PGDB_C031446
DC50-=5.86nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A002071PGDB_C031446PGDB_AS000831View
2D structure for PGDB_C031421
DC50-=3.43nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A002105PGDB_C031421PGDB_AS000831View
2D structure for PGDB_C031434
DC50-=11.82nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A002284PGDB_C031434PGDB_AS000831View
2D structure for PGDB_C031437
DC50-=30.62nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A002352PGDB_C031437PGDB_AS000831View
2D structure for PGDB_C031438
DC50-=9.71nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A002914PGDB_C031438PGDB_AS000831View
2D structure for PGDB_C031431
DC50-=6.67nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A003125PGDB_C031431PGDB_AS000831View
2D structure for PGDB_C031448
DC50-=37.26nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A003376PGDB_C031448PGDB_AS000831View
2D structure for PGDB_C031412
DC50-=15nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A003426PGDB_C031412PGDB_AS000831View
2D structure for PGDB_C031449
DC50-=48.14nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A003654PGDB_C031449PGDB_AS000831View
2D structure for PGDB_C031408
DC50-=89.14nM-—VAV1-293T-VAV1-FLAGWO2026103873A1PGDB_A003954PGDB_C031408PGDB_AS000831View
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