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Cn1cnc(N(c2ccc(-c3cccc(C4CCC(=O)NC4=O)c3Cl)cc2)C2CC2)n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | <= | 20 | nM | - | — | VAV1 | - | - | WO2026114367A1 | PGDB_A001526 | PGDB_C031677 | PGDB_AS000190 | View | |
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primaryT | WO2026114367A1 | PGDB_A078376 | PGDB_C031677 | PGDB_AS002534 | View | |
| IC50 | - | = | 5.09 | nM | - | — | VAV1 | - | - | WO2026114367A1 | PGDB_A079747 | PGDB_C031677 | PGDB_AS000533 | View | |
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primary T cells | WO2026114367A1 | PGDB_A080354 | PGDB_C031677 | PGDB_AS000754 | View | |
| DC50 | - | <= | 20 | nM | - | — | VAV1 | - | primary_human_blood | WO2026114367A1 | PGDB_A081288 | PGDB_C031677 | PGDB_AS001692 | View | |
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primaryT | WO2026114367A1 | PGDB_A081567 | PGDB_C031677 | PGDB_AS000152 | View |