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SIMM · NJU
Assay
PGDB_AS000190
System: cell_based
Target: VAV1
Assay context summary
Assay context
63 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
VAV1
E3
Not specified
Organism
Homo sapiens
Technology
flow_cytometry
Detection target
protein_degradation
Activity compounds and values
Activity records
63 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A000391
PGDB_C031674
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A000437
PGDB_C031732
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A000563
PGDB_C031694
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A000649
PGDB_C031680
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A000675
PGDB_C031717
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A001054
PGDB_C031703
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A001151
PGDB_C031700
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A001387
PGDB_C031698
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A001526
PGDB_C031677
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A001552
PGDB_C031678
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A001701
PGDB_C031701
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A001836
PGDB_C031709
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A002322
PGDB_C031712
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A002475
PGDB_C031690
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A002497
PGDB_C031715
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A002694
PGDB_C031684
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A002696
PGDB_C031716
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A002731
PGDB_C031722
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A002792
PGDB_C031723
PGDB_AS000190
View
DC50
-
<=
20
nM
-
—
VAV1
-
-
WO2026114367A1
PGDB_A002968
PGDB_C031675
PGDB_AS000190
View