Assay
PGDB_AS000032
System: cell_basedCell line: Hep3B2.7-1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-500 | nM | - | — | ESR1 | - | Hep3B2.7-1 | CN116239566A | PGDB_A014168 | PGDB_C019594 | PGDB_AS000032 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ESR1 | - | Hep3B2.7-1 | CN116239566A | PGDB_A029153 | PGDB_C025822 | PGDB_AS000032 | View | |
| IC50 | - | > | 10000 | nM | - | — | ESR1 | - | Hep3B2.7-1 | CN116239566A | PGDB_A037856 | PGDB_C025816 | PGDB_AS000032 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | Hep3B2.7-1 | CN116239566A | PGDB_A074282 | PGDB_C025818 | PGDB_AS000032 | View |