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CC/C(=C(\c1ccc(O)cc1)c1ccc(N2CCN(Cc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)cc1)c1ccc(O)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A007820 | PGDB_C019594 | PGDB_AS001305 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | HCC827 | CN116239566A | PGDB_A012351 | PGDB_C019594 | PGDB_AS001534 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ESR1 | - | Hep3B2.7-1 | CN116239566A | PGDB_A014168 | PGDB_C019594 | PGDB_AS000032 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | Mino | CN116239566A | PGDB_A040247 | PGDB_C019594 | PGDB_AS001392 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MM.1S | CN116239566A | PGDB_A042040 | PGDB_C019594 | PGDB_AS001148 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | T47D | CN116239566A | PGDB_A046415 | PGDB_C019594 | PGDB_AS000239 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A051503 | PGDB_C019594 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | Kasumi-1 | CN116239566A | PGDB_A055854 | PGDB_C019594 | PGDB_AS000517 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SU-DHL-6 | CN116239566A | PGDB_A073532 | PGDB_C019594 | PGDB_AS002532 | View |