Assay
PGDB_AS000104
System: cell_basedCell line: HPAC
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1.031 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A013285 | PGDB_C011632 | PGDB_AS000104 | View | |
| IC50 | - | = | 0.442 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A027057 | PGDB_C011603 | PGDB_AS000104 | View | |
| IC50 | - | = | 1.361 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A028032 | PGDB_C011631 | PGDB_AS000104 | View | |
| IC50 | - | = | 1.043 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A032553 | PGDB_C011633 | PGDB_AS000104 | View | |
| IC50 | - | = | 0.3929 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A065994 | PGDB_C011604 | PGDB_AS000104 | View | |
| IC50 | - | = | 7.253 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A067166 | PGDB_C011587 | PGDB_AS000104 | View | |
| IC50 | - | = | 0.1301 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A074636 | PGDB_C011605 | PGDB_AS000104 | View |