Assay context summary

Assay context

31 activity records
Activity compounds and values

Activity records

31 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007066
IC50-=966.8nM-PDE3A--CN120265631APGDB_A007391PGDB_C007066PGDB_AS000140View
2D structure for PGDB_C007106
IC50-=212.7nM-PDE3A--CN120265631APGDB_A008548PGDB_C007106PGDB_AS000140View
2D structure for PGDB_C007107
IC50-=1125nM-PDE3A--CN120265631APGDB_A010313PGDB_C007107PGDB_AS000140View
2D structure for PGDB_C007124
IC50-=19.16nM-PDE3A--CN120265631APGDB_A013809PGDB_C007124PGDB_AS000140View
2D structure for PGDB_C007133
IC50-=9.48nM-PDE3A--CN120265631APGDB_A015110PGDB_C007133PGDB_AS000140View
2D structure for PGDB_C007080
IC50-=29.35nM-PDE3A--CN120265631APGDB_A015437PGDB_C007080PGDB_AS000140View
2D structure for PGDB_C007100
IC50-=21.77nM-PDE3A--CN120265631APGDB_A017410PGDB_C007100PGDB_AS000140View
2D structure for PGDB_C007148
IC50-=0.87nM-PDE3A--CN120265631APGDB_A017749PGDB_C007148PGDB_AS000140View
2D structure for PGDB_C007147
IC50-=3.7nM-PDE3A--CN120265631APGDB_A018208PGDB_C007147PGDB_AS000140View
2D structure for PGDB_C007104
IC50-=12.3nM-PDE3A--CN120265631APGDB_A018336PGDB_C007104PGDB_AS000140View
2D structure for PGDB_C007093
IC50-=157.83nM-PDE3A--CN120265631APGDB_A019790PGDB_C007093PGDB_AS000140View
2D structure for PGDB_C007140
IC50-=3.1nM-PDE3A--CN120265631APGDB_A023207PGDB_C007140PGDB_AS000140View
2D structure for PGDB_C007116
IC50-=1.6nM-PDE3A--CN120265631APGDB_A024753PGDB_C007116PGDB_AS000140View
2D structure for PGDB_C007092
IC50-=353nM-PDE3A--CN120265631APGDB_A025184PGDB_C007092PGDB_AS000140View
2D structure for PGDB_C007084
IC50-=4.1nM-PDE3A--CN120265631APGDB_A028281PGDB_C007084PGDB_AS000140View
2D structure for PGDB_C007122
IC50-=3.03nM-PDE3A--CN120265631APGDB_A031726PGDB_C007122PGDB_AS000140View
2D structure for PGDB_C007101
IC50-=4.1nM-PDE3A--CN120265631APGDB_A033991PGDB_C007101PGDB_AS000140View
2D structure for PGDB_C007091
IC50-=252.8nM-PDE3A--CN120265631APGDB_A041944PGDB_C007091PGDB_AS000140View
2D structure for PGDB_C007128
IC50-=8.79nM-PDE3A--CN120265631APGDB_A046115PGDB_C007128PGDB_AS000140View
2D structure for PGDB_C007083
IC50-=3.7nM-PDE3A--CN120265631APGDB_A048251PGDB_C007083PGDB_AS000140View