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SIMM · NJU
Assay
PGDB_AS000140
System: cell_based
Target: PDE3A
Assay context summary
Assay context
31 activity records
Assay family
biochemical
System
cell_based
Readout
IC50
Target
PDE3A
E3
Not specified
Activity compounds and values
Activity records
31 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
966.8
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A007391
PGDB_C007066
PGDB_AS000140
View
IC50
-
=
212.7
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A008548
PGDB_C007106
PGDB_AS000140
View
IC50
-
=
1125
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A010313
PGDB_C007107
PGDB_AS000140
View
IC50
-
=
19.16
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A013809
PGDB_C007124
PGDB_AS000140
View
IC50
-
=
9.48
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A015110
PGDB_C007133
PGDB_AS000140
View
IC50
-
=
29.35
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A015437
PGDB_C007080
PGDB_AS000140
View
IC50
-
=
21.77
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A017410
PGDB_C007100
PGDB_AS000140
View
IC50
-
=
0.87
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A017749
PGDB_C007148
PGDB_AS000140
View
IC50
-
=
3.7
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A018208
PGDB_C007147
PGDB_AS000140
View
IC50
-
=
12.3
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A018336
PGDB_C007104
PGDB_AS000140
View
IC50
-
=
157.83
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A019790
PGDB_C007093
PGDB_AS000140
View
IC50
-
=
3.1
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A023207
PGDB_C007140
PGDB_AS000140
View
IC50
-
=
1.6
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A024753
PGDB_C007116
PGDB_AS000140
View
IC50
-
=
353
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A025184
PGDB_C007092
PGDB_AS000140
View
IC50
-
=
4.1
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A028281
PGDB_C007084
PGDB_AS000140
View
IC50
-
=
3.03
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A031726
PGDB_C007122
PGDB_AS000140
View
IC50
-
=
4.1
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A033991
PGDB_C007101
PGDB_AS000140
View
IC50
-
=
252.8
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A041944
PGDB_C007091
PGDB_AS000140
View
IC50
-
=
8.79
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A046115
PGDB_C007128
PGDB_AS000140
View
IC50
-
=
3.7
nM
-
—
PDE3A
-
-
CN120265631A
PGDB_A048251
PGDB_C007083
PGDB_AS000140
View