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O=c1[nH]c2cc3c(Cl)c(-c4cnn(C(F)F)c4Cl)ccc3nc2[nH]1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.87 | nM | - | — | PDE3A | - | - | CN120265631A | PGDB_A017749 | PGDB_C007148 | PGDB_AS000140 | View | |
| IC50 | - | = | 0.09 | nM | - | — | PDE3A | - | SK-MEL-3 | CN120265631A | PGDB_A037941 | PGDB_C007148 | PGDB_AS001659 | View | |
| IC50 | - | = | 0.9 | nM | - | — | PDE3A | - | A2058 | CN120265631A | PGDB_A068145 | PGDB_C007148 | PGDB_AS000265 | View |