Assay
PGDB_AS000150
System: cell_basedCell line: CCRF-CEM
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A013090 | PGDB_C025826 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A018027 | PGDB_C025818 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A032243 | PGDB_C025824 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A048080 | PGDB_C019596 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A048432 | PGDB_C019597 | PGDB_AS000150 | View | |
| IC50 | - | > | 10000 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A050310 | PGDB_C025816 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A051503 | PGDB_C019594 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A075728 | PGDB_C025822 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A076195 | PGDB_C025823 | PGDB_AS000150 | View |