Assay

PGDB_AS000357

System: cell_basedTarget: GSPT1Cell line: HEK293
Assay context summary

Assay context

87 activity records
Assay family% Degradation
Systemcell_based
ReadoutIC50
TargetGSPT1
E3CRBN
Cell lineHEK293
Technologyluminescence
Activity compounds and values

Activity records

87 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008126
IC50-=1uM-—GSPT1CRBNHEK293WO2025043225PGDB_A007083PGDB_C008126PGDB_AS000357View
2D structure for PGDB_C008072
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A008633PGDB_C008072PGDB_AS000357View
2D structure for PGDB_C008069
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A008689PGDB_C008069PGDB_AS000357View
2D structure for PGDB_C008075
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A009591PGDB_C008075PGDB_AS000357View
2D structure for PGDB_C008062
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A010424PGDB_C008062PGDB_AS000357View
2D structure for PGDB_C008059
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A010428PGDB_C008059PGDB_AS000357View
2D structure for PGDB_C008104
IC50-=1uM-—GSPT1CRBNHEK293WO2025043225PGDB_A011001PGDB_C008104PGDB_AS000357View
2D structure for PGDB_C008068
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A011609PGDB_C008068PGDB_AS000357View
2D structure for PGDB_C008058
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A012252PGDB_C008058PGDB_AS000357View
2D structure for PGDB_C008113
IC50-=1uM-—GSPT1CRBNHEK293WO2025043225PGDB_A013049PGDB_C008113PGDB_AS000357View
2D structure for PGDB_C008119
IC50-=1uM-—GSPT1CRBNHEK293WO2025043225PGDB_A013917PGDB_C008119PGDB_AS000357View
2D structure for PGDB_C008046
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A014703PGDB_C008046PGDB_AS000357View
2D structure for PGDB_C008063
IC50-=6uM-—GSPT1CRBNHEK293WO2025043225PGDB_A016708PGDB_C008063PGDB_AS000357View
2D structure for PGDB_C008061
IC50-=3.2uM-—GSPT1CRBNHEK293WO2025043225PGDB_A018384PGDB_C008061PGDB_AS000357View
2D structure for PGDB_C008070
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A018736PGDB_C008070PGDB_AS000357View
2D structure for PGDB_C008121
IC50-=1uM-—GSPT1CRBNHEK293WO2025043225PGDB_A021430PGDB_C008121PGDB_AS000357View
2D structure for PGDB_C008103
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A021812PGDB_C008103PGDB_AS000357View
2D structure for PGDB_C008125
IC50-=1uM-—GSPT1CRBNHEK293WO2025043225PGDB_A025668PGDB_C008125PGDB_AS000357View
2D structure for PGDB_C008086
IC50-=10uM-—GSPT1CRBNHEK293WO2025043225PGDB_A026973PGDB_C008086PGDB_AS000357View
2D structure for PGDB_C008102
IC50-=7uM-—GSPT1CRBNHEK293WO2025043225PGDB_A027010PGDB_C008102PGDB_AS000357View
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