Assay context summary

Assay context

50 activity records
Activity compounds and values

Activity records

50 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007982
Dmax-=4.4%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A008447PGDB_C007982PGDB_AS000429View
2D structure for PGDB_C007979
Dmax-=0.71%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A009108PGDB_C007979PGDB_AS000429View
2D structure for PGDB_C007994
Dmax-=2.5%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A015107PGDB_C007994PGDB_AS000429View
2D structure for PGDB_C008002
Dmax-=1.4%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A015694PGDB_C008002PGDB_AS000429View
2D structure for PGDB_C007981
Dmax-=5%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A016422PGDB_C007981PGDB_AS000429View
2D structure for PGDB_C007988
Dmax-=13%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A018120PGDB_C007988PGDB_AS000429View
2D structure for PGDB_C007980
Dmax-=0.25%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A018925PGDB_C007980PGDB_AS000429View
2D structure for PGDB_C008015
Dmax-=1.4%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A019503PGDB_C008015PGDB_AS000429View
2D structure for PGDB_C007984
Dmax-=0.84%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A020656PGDB_C007984PGDB_AS000429View
2D structure for PGDB_C008006
Dmax-=2.9%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A020752PGDB_C008006PGDB_AS000429View
2D structure for PGDB_C007974
Dmax-=0.99%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A020934PGDB_C007974PGDB_AS000429View
2D structure for PGDB_C007985
Dmax-=3.2%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A021764PGDB_C007985PGDB_AS000429View
2D structure for PGDB_C007971
Dmax-=0.12%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A022075PGDB_C007971PGDB_AS000429View
2D structure for PGDB_C008010
Dmax-=3.7%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A026747PGDB_C008010PGDB_AS000429View
2D structure for PGDB_C007993
Dmax-=5.8%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A030854PGDB_C007993PGDB_AS000429View
2D structure for PGDB_C007990
Dmax-=0.54%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A036915PGDB_C007990PGDB_AS000429View
2D structure for PGDB_C007975
Dmax-=1.2%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A040527PGDB_C007975PGDB_AS000429View
2D structure for PGDB_C007997
Dmax-=0.14%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A040707PGDB_C007997PGDB_AS000429View
2D structure for PGDB_C007989
Dmax-=3.3%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A041448PGDB_C007989PGDB_AS000429View
2D structure for PGDB_C008005
Dmax-=0.83%10 uM6 hGSPT1-HEK293WO2025043225PGDB_A043168PGDB_C008005PGDB_AS000429View