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SIMM · NJU
Assay
PGDB_AS000429
System: cell_based
Target: GSPT1
Cell line: HEK293
Assay context summary
Assay context
50 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
GSPT1
E3
Not specified
Cell line
HEK293
Activity compounds and values
Activity records
50 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
4.4
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A008447
PGDB_C007982
PGDB_AS000429
View
Dmax
-
=
0.71
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A009108
PGDB_C007979
PGDB_AS000429
View
Dmax
-
=
2.5
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A015107
PGDB_C007994
PGDB_AS000429
View
Dmax
-
=
1.4
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A015694
PGDB_C008002
PGDB_AS000429
View
Dmax
-
=
5
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A016422
PGDB_C007981
PGDB_AS000429
View
Dmax
-
=
13
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A018120
PGDB_C007988
PGDB_AS000429
View
Dmax
-
=
0.25
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A018925
PGDB_C007980
PGDB_AS000429
View
Dmax
-
=
1.4
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A019503
PGDB_C008015
PGDB_AS000429
View
Dmax
-
=
0.84
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A020656
PGDB_C007984
PGDB_AS000429
View
Dmax
-
=
2.9
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A020752
PGDB_C008006
PGDB_AS000429
View
Dmax
-
=
0.99
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A020934
PGDB_C007974
PGDB_AS000429
View
Dmax
-
=
3.2
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A021764
PGDB_C007985
PGDB_AS000429
View
Dmax
-
=
0.12
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A022075
PGDB_C007971
PGDB_AS000429
View
Dmax
-
=
3.7
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A026747
PGDB_C008010
PGDB_AS000429
View
Dmax
-
=
5.8
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A030854
PGDB_C007993
PGDB_AS000429
View
Dmax
-
=
0.54
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A036915
PGDB_C007990
PGDB_AS000429
View
Dmax
-
=
1.2
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A040527
PGDB_C007975
PGDB_AS000429
View
Dmax
-
=
0.14
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A040707
PGDB_C007997
PGDB_AS000429
View
Dmax
-
=
3.3
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A041448
PGDB_C007989
PGDB_AS000429
View
Dmax
-
=
0.83
%
10 uM
6 h
GSPT1
-
HEK293
WO2025043225
PGDB_A043168
PGDB_C008005
PGDB_AS000429
View